Abstract
The Concise Guide to PHARMACOLOGY 2021/22 is the fifth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of nearly 1900 human drug targets with an emphasis on selective pharmacology (where available), plus links to the open access knowledgebase source of drug targets and their ligands (www.guidetopharmacology.org), which provides more detailed views of target and ligand properties. Although the Concise Guide constitutes over 500 pages, the material presented is substantially reduced compared to information and links presented on the website. It provides a permanent, citable, point-in-time record that will survive database updates. The full contents of this section can be found at http://onlinelibrary.wiley.com/doi/bph.15538. G protein-coupled receptors are one of the six major pharmacological targets into which the Guide is divided, with the others being: ion channels, nuclear hormone receptors, catalytic receptors, enzymes and transporters. These are presented with nomenclature guidance and summary information on the best available pharmacological tools, alongside key references and suggestions for further reading. The landscape format of the Concise Guide is designed to facilitate comparison of related targets from material contemporary to mid-2021, and supersedes data presented in the 2019/20, 2017/18, 2015/16 and 2013/14 Concise Guides and previous Guides to Receptors and Channels. It is produced in close conjunction with the Nomenclature and Standards Committee of the International Union of Basic and Clinical Pharmacology (NC-IUPHAR), therefore, providing official IUPHAR classification and nomenclature for human drug targets, where appropriate.
| Original language | English |
|---|---|
| Pages (from-to) | S27-S156 |
| Number of pages | 130 |
| Journal | British Journal of Pharmacology |
| Volume | 178 |
| Issue number | S1 |
| DOIs | |
| Publication status | Published - Oct 2021 |
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In: British Journal of Pharmacology, Vol. 178, No. S1, 10.2021, p. S27-S156.
Research output: Contribution to journal › Article › Other › peer-review
TY - JOUR
T1 - THE CONCISE GUIDE TO PHARMACOLOGY 2021/22
T2 - G protein-coupled receptors
AU - Alexander, Stephen P.H.
AU - Christopoulos, Arthur
AU - Davenport, Anthony P.
AU - Kelly, Eamonn
AU - Mathie, Alistair
AU - Peters, John A.
AU - Veale, Emma L.
AU - Armstrong, Jane F.
AU - Faccenda, Elena
AU - Harding, Simon D.
AU - Pawson, Adam J.
AU - Southan, Christopher
AU - Davies, Jamie A.
AU - Abbracchio, Maria Pia
AU - Alexander, Wayne
AU - Al-hosaini, Khaled
AU - Bäck, Magnus
AU - Barnes, Nicholas M.
AU - Bathgate, Ross
AU - Beaulieu, Jean Martin
AU - Bernstein, Kenneth E.
AU - Bettler, Bernhard
AU - Birdsall, Nigel J.M.
AU - Blaho, Victoria
AU - Boulay, Francois
AU - Bousquet, Corinne
AU - Bräuner-Osborne, Hans
AU - Burnstock, Geoffrey
AU - Caló, Girolamo
AU - Castaño, Justo P.
AU - Catt, Kevin J.
AU - Ceruti, Stefania
AU - Chazot, Paul
AU - Chiang, Nan
AU - Chini, Bice
AU - Chun, Jerold
AU - Cianciulli, Antonia
AU - Civelli, Olivier
AU - Clapp, Lucie H.
AU - Couture, Réjean
AU - Csaba, Zsolt
AU - Dahlgren, Claes
AU - Dent, Gordon
AU - Singh, Khuraijam Dhanachandra
AU - Douglas, Steven D.
AU - Dournaud, Pascal
AU - Eguchi, Satoru
AU - Escher, Emanuel
AU - Filardo, Edward J.
AU - Fong, Tung
AU - Fumagalli, Marta
AU - Gainetdinov, Raul R.
AU - Gasparo, Marc de
AU - Gerard, Craig
AU - Gershengorn, Marvin
AU - Gobeil, Fernand
AU - Goodfriend, Theodore L.
AU - Goudet, Cyril
AU - Gregory, Karen J.
AU - Gundlach, Andrew L.
AU - Hamann, Jörg
AU - Hanson, Julien
AU - Hauger, Richard L.
AU - Hay, Debbie L.
AU - Heinemann, Akos
AU - Hollenberg, Morley D.
AU - Holliday, Nicholas D.
AU - Horiuchi, Mastgugu
AU - Hoyer, Daniel
AU - Hunyady, László
AU - Husain, Ahsan
AU - IJzerman, Adriaan P.
AU - Inagami, Tadashi
AU - Jacobson, Kenneth A.
AU - Jensen, Robert T.
AU - Jockers, Ralf
AU - Jonnalagadda, Deepa
AU - Karnik, Sadashiva
AU - Kaupmann, Klemens
AU - Kemp, Jacqueline
AU - Kennedy, Charles
AU - Kihara, Yasuyuki
AU - Kitazawa, Takio
AU - Kozielewicz, Pawel
AU - Kreienkamp, Hans Jürgen
AU - Kukkonen, Jyrki P.
AU - Langenhan, Tobias
AU - Leach, Katie
AU - Lecca, Davide
AU - Lee, John D.
AU - Leeman, Susan E.
AU - Leprince, Jérôme
AU - Li, Xaria X.
AU - Williams, Tom Lloyd
AU - Lolait, Stephen J.
AU - Lupp, Amelie
AU - Macrae, Robyn
AU - Maguire, Janet
AU - Mazella, Jean
AU - McArdle, Craig A.
AU - Melmed, Shlomo
AU - Michel, Martin C.
AU - Miller, Laurence J.
AU - Mitolo, Vincenzo
AU - Mouillac, Bernard
AU - Müller, Christa E.
AU - Murphy, Philip
AU - Nahon, Jean Louis
AU - Ngo, Tony
AU - Norel, Xavier
AU - Nyimanu, Duuamene
AU - O’Carroll, Anne Marie
AU - Offermanns, Stefan
AU - Panaro, Maria Antonietta
AU - Parmentier, Marc
AU - Pertwee, Roger G.
AU - Pin, Jean Philippe
AU - Prossnitz, Eric R.
AU - Quinn, Mark
AU - Ramachandran, Rithwik
AU - Ray, Manisha
AU - Reinscheid, Rainer K.
AU - Rondard, Philippe
AU - Rovati, G. Enrico
AU - Ruzza, Chiara
AU - Sanger, Gareth J.
AU - Schöneberg, Torsten
AU - Schulte, Gunnar
AU - Schulz, Stefan
AU - Segaloff, Deborah L.
AU - Serhan, Charles N.
AU - Stoddart, Leigh A.
AU - Sugimoto, Yukihiko
AU - Summers, Roger
AU - Tan, Valerie P.
AU - Thal, David
AU - Thomas, Walter
AU - Timmermans, Pieter B.M.W.M.
AU - Tirupula, Kalyan
AU - Tulipano, Giovanni
AU - Unal, Hamiyet
AU - Unger, Thomas
AU - Valant, Celine
AU - Vanderheyden, Patrick
AU - Vaudry, David
AU - Vaudry, Hubert
AU - Vilardaga, Jean Pierre
AU - Walker, Christopher S.
AU - Wang, Ji Ming
AU - Ward, Donald T.
AU - Wester, Hans Jürgen
AU - Willars, Gary B.
AU - Woodruff, Trent M.
AU - Yao, Chengcan
AU - Ye, Richard D.
N1 - Publisher Copyright: © 2021 The Authors. British Journal of Pharmacology published by John Wiley & Sons Ltd on behalf of The British Pharmacological Society Copyright: Copyright 2021 Elsevier B.V., All rights reserved.
PY - 2021/10
Y1 - 2021/10
N2 - The Concise Guide to PHARMACOLOGY 2021/22 is the fifth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of nearly 1900 human drug targets with an emphasis on selective pharmacology (where available), plus links to the open access knowledgebase source of drug targets and their ligands (www.guidetopharmacology.org), which provides more detailed views of target and ligand properties. Although the Concise Guide constitutes over 500 pages, the material presented is substantially reduced compared to information and links presented on the website. It provides a permanent, citable, point-in-time record that will survive database updates. The full contents of this section can be found at http://onlinelibrary.wiley.com/doi/bph.15538. G protein-coupled receptors are one of the six major pharmacological targets into which the Guide is divided, with the others being: ion channels, nuclear hormone receptors, catalytic receptors, enzymes and transporters. These are presented with nomenclature guidance and summary information on the best available pharmacological tools, alongside key references and suggestions for further reading. The landscape format of the Concise Guide is designed to facilitate comparison of related targets from material contemporary to mid-2021, and supersedes data presented in the 2019/20, 2017/18, 2015/16 and 2013/14 Concise Guides and previous Guides to Receptors and Channels. It is produced in close conjunction with the Nomenclature and Standards Committee of the International Union of Basic and Clinical Pharmacology (NC-IUPHAR), therefore, providing official IUPHAR classification and nomenclature for human drug targets, where appropriate.
AB - The Concise Guide to PHARMACOLOGY 2021/22 is the fifth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of nearly 1900 human drug targets with an emphasis on selective pharmacology (where available), plus links to the open access knowledgebase source of drug targets and their ligands (www.guidetopharmacology.org), which provides more detailed views of target and ligand properties. Although the Concise Guide constitutes over 500 pages, the material presented is substantially reduced compared to information and links presented on the website. It provides a permanent, citable, point-in-time record that will survive database updates. The full contents of this section can be found at http://onlinelibrary.wiley.com/doi/bph.15538. G protein-coupled receptors are one of the six major pharmacological targets into which the Guide is divided, with the others being: ion channels, nuclear hormone receptors, catalytic receptors, enzymes and transporters. These are presented with nomenclature guidance and summary information on the best available pharmacological tools, alongside key references and suggestions for further reading. The landscape format of the Concise Guide is designed to facilitate comparison of related targets from material contemporary to mid-2021, and supersedes data presented in the 2019/20, 2017/18, 2015/16 and 2013/14 Concise Guides and previous Guides to Receptors and Channels. It is produced in close conjunction with the Nomenclature and Standards Committee of the International Union of Basic and Clinical Pharmacology (NC-IUPHAR), therefore, providing official IUPHAR classification and nomenclature for human drug targets, where appropriate.
UR - http://www.scopus.com/inward/record.url?scp=85115083018&partnerID=8YFLogxK
U2 - 10.1111/bph.15538
DO - 10.1111/bph.15538
M3 - Article
AN - SCOPUS:85115083018
SN - 1476-5381
VL - 178
SP - S27-S156
JO - British Journal of Pharmacology
JF - British Journal of Pharmacology
IS - S1
ER -