Synthesis of 2-substituted 3-acylbenzo[b]furans via the palladium catalysed carbonylative cyclisation of ortho-hydroxytolans

Henning Lütjens, Peter J. Scammells

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Abstract

A palladium-catalysed cyclisation with concomitant carbonylation via insertion of carbon monoxide was used to prepare several potential adenosine antagonists possessing a benzo[b]furan skeleton with a formyl group in the 3-position.
Original languageEnglish
Pages (from-to)1079-1081
Number of pages3
JournalSynlett
Issue number7
DOIs
Publication statusPublished - 1 Jan 1999

Keywords

  • Adenosine antagonist
  • Benzofuran
  • Carbonylative cyclisation
  • Palladium

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