Parasiticidal 2-alkoxy- and 2-aryloxyiminoalkyl trifluoromethanesulfonanilides

Abdelselam Ali; Timothy M. Altamore; Marianne Bliese; Petr Fisara; Andris J. Liepa; Adam G. Meyer; Oahn Nguyen; Roger M. Sargent; David G. Sawutz; David A. Winkler; Kevin N. Winzenberg; Angela Ziebell

doi:10.1016/j.bmcl.2007.10.090

Parasiticidal 2-alkoxy- and 2-aryloxyiminoalkyl trifluoromethanesulfonanilides

Abdelselam Ali
, Timothy M. Altamore
, Marianne Bliese
, Petr Fisara
, Andris J. Liepa
, Adam G. Meyer
, Oahn Nguyen
, Roger M. Sargent
, David G. Sawutz
, David A. Winkler
, Kevin N. Winzenberg
, Angela Ziebell

Research output: Contribution to journal › Article › Other

11 Citations (Scopus)

Abstract

A series of novel 2-alkoxy- and 2-aryloxyiminoalkyl trifluoromethanesulfonanilide derivatives have shown significant in vitro parasiticidal activity against the ectoparasites Ctenocephalides felis and Rhipicephalus sanguineus. A number of these compounds also displayed significant in vitro endoparasite activity against the nematode Haemonchus contortus.

Original language	English
Pages (from-to)	252-255
Number of pages	4
Journal	Bioorganic and Medicinal Chemistry Letters
Volume	18
Issue number	1
DOIs	https://doi.org/10.1016/j.bmcl.2007.10.090
Publication status	Published - 1 Jan 2008
Externally published	Yes

Keywords

Ctenocephalides felis (cat flea)
Haemonchus contortus
Oxime ether
Parasiticide
Rhipicephalus sanguineus (brown dog tick)
Trifluoromethanesulfonanilide

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10.1016/j.bmcl.2007.10.090

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title = "Parasiticidal 2-alkoxy- and 2-aryloxyiminoalkyl trifluoromethanesulfonanilides",

abstract = "A series of novel 2-alkoxy- and 2-aryloxyiminoalkyl trifluoromethanesulfonanilide derivatives have shown significant in vitro parasiticidal activity against the ectoparasites Ctenocephalides felis and Rhipicephalus sanguineus. A number of these compounds also displayed significant in vitro endoparasite activity against the nematode Haemonchus contortus. ",

keywords = "Ctenocephalides felis (cat flea), Haemonchus contortus, Oxime ether, Parasiticide, Rhipicephalus sanguineus (brown dog tick), Trifluoromethanesulfonanilide",

author = "Abdelselam Ali and Altamore, \{Timothy M.\} and Marianne Bliese and Petr Fisara and Liepa, \{Andris J.\} and Meyer, \{Adam G.\} and Oahn Nguyen and Sargent, \{Roger M.\} and Sawutz, \{David G.\} and Winkler, \{David A.\} and Winzenberg, \{Kevin N.\} and Angela Ziebell",

year = "2008",

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day = "1",

doi = "10.1016/j.bmcl.2007.10.090",

language = "English",

volume = "18",

pages = "252--255",

journal = "Bioorganic and Medicinal Chemistry Letters",

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TY - JOUR

T1 - Parasiticidal 2-alkoxy- and 2-aryloxyiminoalkyl trifluoromethanesulfonanilides

AU - Ali, Abdelselam

AU - Altamore, Timothy M.

AU - Bliese, Marianne

AU - Fisara, Petr

AU - Liepa, Andris J.

AU - Meyer, Adam G.

AU - Nguyen, Oahn

AU - Sargent, Roger M.

AU - Sawutz, David G.

AU - Winkler, David A.

AU - Winzenberg, Kevin N.

AU - Ziebell, Angela

PY - 2008/1/1

Y1 - 2008/1/1

N2 - A series of novel 2-alkoxy- and 2-aryloxyiminoalkyl trifluoromethanesulfonanilide derivatives have shown significant in vitro parasiticidal activity against the ectoparasites Ctenocephalides felis and Rhipicephalus sanguineus. A number of these compounds also displayed significant in vitro endoparasite activity against the nematode Haemonchus contortus.

AB - A series of novel 2-alkoxy- and 2-aryloxyiminoalkyl trifluoromethanesulfonanilide derivatives have shown significant in vitro parasiticidal activity against the ectoparasites Ctenocephalides felis and Rhipicephalus sanguineus. A number of these compounds also displayed significant in vitro endoparasite activity against the nematode Haemonchus contortus.

KW - Ctenocephalides felis (cat flea)

KW - Haemonchus contortus

KW - Oxime ether

KW - Parasiticide

KW - Rhipicephalus sanguineus (brown dog tick)

KW - Trifluoromethanesulfonanilide

UR - https://www.scopus.com/pages/publications/37549016405

U2 - 10.1016/j.bmcl.2007.10.090

DO - 10.1016/j.bmcl.2007.10.090

M3 - Article

C2 - 18006308

SN - 0960-894X

VL - 18

SP - 252

EP - 255

JO - Bioorganic and Medicinal Chemistry Letters

JF - Bioorganic and Medicinal Chemistry Letters

IS - 1

ER -

Parasiticidal 2-alkoxy- and 2-aryloxyiminoalkyl trifluoromethanesulfonanilides

Abstract

Keywords

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