Drug discovery beyond the rule of 5 - opportunities and challenges

Bradley C. Doak; Jan Kihlberg

doi:10.1080/17460441.2017.1264385

Drug discovery beyond the rule of 5 - opportunities and challenges

Bradley C. Doak, Jan Kihlberg

Medicinal Chemistry

Research output: Contribution to journal › Article › Research › peer-review

91 Citations (Scopus)

Original language	English
Pages (from-to)	115-119
Number of pages	5
Journal	Expert Opinion on Drug Discovery
Volume	12
Issue number	2
DOIs	https://doi.org/10.1080/17460441.2017.1264385
Publication status	Published - 2017

Keywords

Beyond rule of 5
conformational flexibility
difficult target
macrocycle
oral absorption

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10.1080/17460441.2017.1264385

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Drug discovery beyond the rule of 5 - opportunities and challenges

Keywords

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