Aziridination of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate

Jiayin Li; Jiang Lin Liang; Philip Wai Hong Chan; Chi Ming Che

doi:10.1016/j.tetlet.2004.01.127

Aziridination of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate

Jiayin Li
, Jiang Lin Liang
, Philip Wai Hong Chan
, Chi Ming Che

Research output: Contribution to journal › Article › Research › peer-review

87 Citations (Scopus)

Abstract

Aziridination of a variety of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate under mild conditions (K₂CO ₃, CH₂Cl₂) and ambient temperature were achieved in good to excellent yields (up to 99%), and conversions. The practicality and simplicity of this C-N bond formation protocol was exemplified by its application to the aziridination of cholesteryl acetate in a stereoselective manner.

Original language	English
Pages (from-to)	2685-2688
Number of pages	4
Journal	Tetrahedron Letters
Volume	45
Issue number	12
DOIs	https://doi.org/10.1016/j.tetlet.2004.01.127
Publication status	Published - 15 Mar 2004
Externally published	Yes

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10.1016/j.tetlet.2004.01.127

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title = "Aziridination of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate",

abstract = "Aziridination of a variety of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate under mild conditions (K2CO 3, CH2Cl2) and ambient temperature were achieved in good to excellent yields (up to 99\%), and conversions. The practicality and simplicity of this C-N bond formation protocol was exemplified by its application to the aziridination of cholesteryl acetate in a stereoselective manner.",

author = "Jiayin Li and Liang, \{Jiang Lin\} and Chan, \{Philip Wai Hong\} and Che, \{Chi Ming\}",

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T1 - Aziridination of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate

AU - Li, Jiayin

AU - Liang, Jiang Lin

AU - Chan, Philip Wai Hong

AU - Che, Chi Ming

PY - 2004/3/15

Y1 - 2004/3/15

N2 - Aziridination of a variety of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate under mild conditions (K2CO 3, CH2Cl2) and ambient temperature were achieved in good to excellent yields (up to 99%), and conversions. The practicality and simplicity of this C-N bond formation protocol was exemplified by its application to the aziridination of cholesteryl acetate in a stereoselective manner.

AB - Aziridination of a variety of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate under mild conditions (K2CO 3, CH2Cl2) and ambient temperature were achieved in good to excellent yields (up to 99%), and conversions. The practicality and simplicity of this C-N bond formation protocol was exemplified by its application to the aziridination of cholesteryl acetate in a stereoselective manner.

UR - https://www.scopus.com/pages/publications/1542362197

U2 - 10.1016/j.tetlet.2004.01.127

DO - 10.1016/j.tetlet.2004.01.127

M3 - Article

AN - SCOPUS:1542362197

SN - 0040-4039

VL - 45

SP - 2685

EP - 2688

JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 12

ER -

Aziridination of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate

Abstract

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