1,2,4-triazolo[1,5-a][1,3,5]triazines (5-azapurines): synthesis and biological activity

Anton V. Dolzhenko, Anna V. Dolzhenko, Wai Keung Chui

Research output: Contribution to journalArticleResearchpeer-review

50 Citations (Scopus)


The present review gives an account of the various synthetic routes to the 5-aza-analogue of purine-1,2,4-triazolo[1,5-a][1,3,5]triazine nucleus and polyfused systems bearing this heterocyclic core. Data concerning biological activity of the compounds with 1,2,4-triazolo[1,5-a][1,3,5]triazine skeleton are also discussed.{A figure is presented}.

Original languageEnglish
Pages (from-to)1723-1759
Number of pages37
Issue number8
Publication statusPublished - 1 Aug 2006
Externally publishedYes

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