Research Output per year
Research Output 1997 2019
- 1 - 50 out of 117 results
- Publication Year, Title (descending)
2019
Aurone derivatives as Vps34 inhibitors that modulate autophagy
Li, G., Boyle, J. W., Ko, C. N., Zeng, W., Wong, V. K. W., Wan, J. B., Chan, P. W. H., Ma, D. L. & Leung, C. H., 1 Jan 2019, In : Acta Pharmaceutica Sinica B. 9, 3, p. 537–544 8 p.Research output: Contribution to journal › Article › Research › peer-review
Open Access
File
Gold Catalyzed Photoredox C1-Alkynylation of N-Alkyl-1,2,3,4- tetrahydroisoquinolines by 1-Bromoalkynes with UVA LED Light
Zhao, Y., Jin, J. & Chan, P. W. H., 1 Jan 2019, In : Advanced Synthesis and Catalysis. 361, 6, p. 1313-1321 9 p.Research output: Contribution to journal › Article › Research › peer-review
2018
Brønsted acid-catalysed allylic amination of 1-(2-aminoaryl)prop-2-en-1-ols to 1,2-dihydroquinolines
Day, D. P., Henry, S. A., Zhao, Y., Jin, J., Clarkson, G. J. & Chan, P. W. H., 19 Jun 2018, In : Australian Journal of Chemistry. 71, 9, p. 673-681 9 p.Research output: Contribution to journal › Article › Research › peer-review
Chiral Brønsted acid and gold catalyzed enantioselective synthesis of 1,8-dihydroindeno[2,1-b]pyrroles
Jin, J., Zhao, Y., Sze, E. M. L., Kothandaraman, P. & Chan, P. W. H., 21 Dec 2018, In : Advanced Synthesis and Catalysis. 360, 24, p. 4744-4753 10 p.Research output: Contribution to journal › Article › Research › peer-review
Chiral Brønsted acid catalyzed enantioselective dehydrative nazarov-type electrocyclization of aryl and 2-thienyl vinyl alcohols
Jin, J., Zhao, Y., Gouranourimi, A., Ariafard, A. & Chan, P. W. H., 2 May 2018, In : Journal of the American Chemical Society. 140, 17, p. 5834-5841 8 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed double cycloisomerization of 1-ene-4,10-diynyl esters to bicyclo[6.3.0]undeca-2,4,9-trienyl esters
Mathiew, M., Tan, J. K. & Chan, P. W. H., 22 Oct 2018, In : Angewandte Chemie - International Edition. 57, 43, p. 14235-14239 5 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-Catalyzed Formal [4 + 2] Cycloaddition of 5-(Ethynylamino)pent-2-yn-1-yl Esters to 1,2,3,5-Tetrahydrobenzo [g] quinolines
Chen, X., Merrett, J. T. & Hong Chan, P. W., 16 Mar 2018, In : Organic Letters. 20, 6, p. 1542-1545 4 p.Research output: Contribution to journal › Article › Research › peer-review
2017
Brønsted Acid-Mediated Cycloaromatization of 1H-Indol-2-yl Propargyl Benzoates to 7H-Benzo[c]carbazoles
Tan, J. K., Mathiew, M., Nayak, S. & Chan, P. W. H., 4 Jul 2017, In : Chemistry - An Asian Journal. 12, 13, p. 1475-1479 5 p.Research output: Contribution to journal › Article › Research › peer-review
Open Access
File
Brønsted Base-Mediated Aziridination of 2-Alkyl-Substituted-1,3-Dicarbonyl Compounds and 2-Acyl-Substituted-1,4-Dicarbonyl Compounds by Iminoiodanes
Tejo, C., Tirtorahardjo, D., Day, D. P., Ma, D-L. E., Leung, C-H. D. & Chan, P. W. H., 2017, In : Australian Journal of Chemistry. 70, 4, p. 430-435 6 p.Research output: Contribution to journal › Article › Research › peer-review
Open Access
File
Gold-Catalyzed Dehydrogenative Cycloisomerization of 1,4-Enyne Esters to 3,5-Disubstituted Phenol Derivatives
Chen, C., Chen, X., Zhang, X., Wang, S., Rao, W. & Chan, P. W. H., 19 Dec 2017, In : Advanced Synthesis and Catalysis. 359, 24, p. 4359-4368 10 p.Research output: Contribution to journal › Article › Research › peer-review
Silver-Catalyzed 1,3-Acyloxy Migration/Diels-Alder Reaction of 1,9-Dien-4-yne Esters to Partially Hydrogenated Isoquinolines
Zhao, Y., Jin, J., Boyle, J. W., Lee, B. R., Day, D. P., Susanti, D., Clarkson, G. J. & Chan, P. W. H., 17 Mar 2017, In : Journal of Organic Chemistry. 82, 6, p. 2826-2834 9 p.Research output: Contribution to journal › Article › Research › peer-review
2016
Copper-Mediated Cross-Dehydrogenative Coupling of 2-Methylpyridine and 8-Methylquinoline with Methyl Ketones and Benzamides
Kumar, G. S., Boyle, J. W., Tejo, C. & Chan, P. W. H., 4 Feb 2016, In : Chemistry - An Asian Journal. 11, 3, p. 385-389 5 p.Research output: Contribution to journal › Article › Research › peer-review
Gold- and Brønsted Acid-Catalyzed Cycloisomerization of 1,8-Diynyl Vinyl Acetates to Bicyclo[2.2.1]hept-2-en-7-ones
Chen, X., Day, D. P., Teo, W. T. & Chan, P. W. H., 18 Nov 2016, In : Organic Letters. 18, 22, p. 5936-5939 4 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-Catalyzed Aminoalkenylation of β-Amino-1,n-Diynols to Cycloalkyl-, Piperidinyl- and Pyranyl-Fused Pyrroles
Kothandaraman, P., Zhao, Y., Lee, B. R., Le Ng, C. J., Lee, J. Y., Ayers, B. J. & Chan, P. W. H., 28 Apr 2016, In : Advanced Synthesis and Catalysis. 358, 9, p. 1385-1391 7 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-Catalyzed Sequential Cyclization of 1-En-3,9-Diyne Esters to Partially Hydrogenated 3H-Dicyclopenta[a,b]naphthalenes
Rao, W., Boyle, J. W. & Chan, P. W. H., 4 May 2016, In : Chemistry - A European Journal. 22, 19, p. 6532-6536 5 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-Catalyzed Tandem 1,3-Migration/Double Cyclopropanation of 1-Ene-4,n-diyne Esters to Tetracyclodecene and Tetracycloundecene Derivatives
Chen, C., Zou, Y., Chen, X., Zhang, X., Rao, W. & Chan, P. W. H., 16 Sep 2016, In : Organic Letters. 18, 18, p. 4730-4733 4 p.Research output: Contribution to journal › Article › Research › peer-review
Structure-based screening and optimization of cytisine derivatives as inhibitors of the menin-MLL interaction
Zhong, H-J., Lee, B. R., Boyle, J. W., Wang, W., Ma, D-L. E., Hong Chan, P. W. & Leung, C-H. D., 30 Apr 2016, In : Chemical Communications. 52, 34, p. 5788-5791 4 p.Research output: Contribution to journal › Article › Research › peer-review
Synthesis of 1,4-amino alcohols by Grignard reagent addition to THF and N-tosyliminobenzyliodinane
Tejo, C., See, Y. F. A., Mathiew, M. & Chan, P. W. H., 2016, In : Organic and Biomolecular Chemistry. 14, 3, p. 844-848 5 p.Research output: Contribution to journal › Article › Research › peer-review
2015
A label-free G-quadruplex-based mercury detection assay employing the exonuclease III-mediated cleavage of T-Hg2+-T mismatched DNA
Wang, W., Kang, T-S., Chan, P. W. H., Lu, J-J., Chen, X-P., Leung, C-H. D. & Ma, D-L. E., 2015, In : Science and Technology of Advanced Materials. 16, 6, p. 1-6 6 p.Research output: Contribution to journal › Article › Research › peer-review
Open Access
File
Crystal structure of (Z)-1-phenyl-3-styrylundeca-2-en-4, 10-diyn-1-ol
Ganguly, R., Sally, U. & Chan, P. W. H., 2015, In : Acta Crystallographica Section E: Structure Reports Online. 71, 1, p. 64 - 64 1 p.Research output: Contribution to journal › Article › Other › peer-review
Open Access
File
Discovery of a small-molecule inhibitor of STAT3 by ligand-based pharmacophore screening
Leung, K-H., Liu, L-J., Lin, S., Lu, L., Zhong, H-J., Susanti, D., Rao, W., Wang, M., Che, W. I., Chan, D. S-H., Leung, C-H. D., Chan, P. W. H. & Ma, D-L. E., 2015, In : Methods. 71, C, p. 38-43 6 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed cycloisomerization and Diels-Alder reaction of 1,4,9-dienyne esters to 3 a,6-methanoisoindole esters with pro-inflammatory cytokine antagonist activity
Susanti, D., Liu, L-J., Rao, W., Lin, S., Ma, D-L. E., Leung, C-H. D. & Chan, P. W. H., 2015, In : Chemistry - A European Journal. 21, 25, p. 9111-9118 8 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed cycloisomerization and Diels-Alder reaction of 1,6-diyne esters with alkenes and diazenes to hydronaphthalenes and -cinnolines
Yan, J., Tay, G. L., Neo, C., Lee, B. R. & Chan, P. W. H., 2015, In : Organic Letters. 17, 17, p. 4176-4179 4 p.Research output: Contribution to journal › Article › Research › peer-review
Harnessing the versatile reactivity of propargyl alcohols and their derivatives for sustainable complex molecule synthesis
Ayers, B. J. & Chan, P. W. H., 2015, In : Synlett. 26, 10, p. 1305-1339 35 p.Research output: Contribution to journal › Article › Research › peer-review
Iminoiodane- and Bronsted base-mediated cross dehydrogenative coupling of cyclic ethers with 1,3-dicarbonyl compounds
Tejo, C., Sim, X. R., Lee, B. R., Ayers, B. J., Leung, C-H. D., Ma, D-L. E. & Chan, P. W. H., 2015, In : Molecules. 20, 7, p. 13336-13353 18 p.Research output: Contribution to journal › Article › Research › peer-review
Open Access
Ligand-controlled product selectivity in gold-catalyzed double cycloisomerization of 1,11-dien-3,9-diyne benzoates
Rao, W., Susanti, D., Ayers, B. J. & Chan, P. W. H., 2015, In : Journal of the American Chemical Society. 137, 19, p. 6350-6355 6 p.Research output: Contribution to journal › Article › Research › peer-review
Pharmacophore modeling for the identification of small-molecule inhibitors of TACE
Liu, L-J., Leung, K-H., Lin, S., Chan, D. S-H., Susanti, D., Rao, W., Chan, P. W. H., Ma, D-L. E. & Leung, C-H. D., 2015, In : Methods. 71, p. 92 - 97 6 p.Research output: Contribution to journal › Article › Research › peer-review
Silver Triflate Catalyzed Cyclopropyl Carbinol Rearrangement for Benzo[b]oxepine and 2H-Chromene Synthesis
Chan, P. W. H., Teo, W. T., Koh, S. W. Y., Lee, B. R., Ayers, B. J., Ma, D-L. E. & Leung, C-H. D., 1 Jul 2015, In : European Journal of Organic Chemistry. 2015, 20, p. 4447-4456 10 p.Research output: Contribution to journal › Article › Research › peer-review
2014
A G-quadruplex-based platform for the detection of Hg2+ ions using a luminescent iridium(III) complex
Lin, S., He, B., Chan, D. S-H., Chan, P. W. H., Leung, C-H. D. & Ma, D-L. E., 2014, In : RSC Advances. 4, 97, p. 54826 - 54831 6 p.Research output: Contribution to journal › Article › Research › peer-review
Open Access
File
Bronsted acid catalyzed amination of 1,3-dicarbonyl compounds by iminoiodanes
Tejo, C., Yeo, H. Q. & Chan, P. W. H., 2014, In : Synlett. 25, 2, p. 201 - 204 4 p.Research output: Contribution to journal › Article › Other › peer-review
Discovery of a natural product-like iNOS inhibitor by molecular docking with potential neuroprotective effects in vivo
Zhong, H-J., Liu, L-J., Chong, C-M., Lu, L., Wang, M., Chan, D. S-H., Chan, P. W. H., Lee, S. M-Y., Ma, D-L. E. & Leung, C-H. D., 2014, In : PLoS ONE. 9, 4, p. 1-10 10 p., e92905.Research output: Contribution to journal › Article › Research › peer-review
Open Access
File
Gold-catalyzed [2+2+1] cycloaddition of 1,6-diyne carbonates and esters with aldehydes to 4-(cyclohexa-1,3-dienyl)-1,3-dioxolanes
Rao, W. & Chan, P. W. H., 2014, In : Chemistry - A European Journal. 20, 3, p. 713 - 718 6 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed benzannulation of 5-hydroxy-3-oxoalk-6-ynoate esters to o-phenolic esters
Teo, W. T., Rao, W., Ng, C. J. H., Koh, S. W. Y. & Chan, P. W. H., 2014, In : Organic Letters. 16, 4, p. 1248 - 1251 4 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed cycloisomerization of 1,6,8-dienyne carbonates and esters to cis-cyclohepta-4,8-diene-fused pyrrolidines
Rao, W., Sally, Berry, S. N. & Chan, P. W. H., 2014, In : Chemistry - A European Journal. 20, 41, p. 13174 - 13180 7 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed cycloisomerization of 1,6-diyne esters to 1H-cyclopenta[b]naphthalenes, cis-cyclopenten-2-yl delta-diketones, and bicyclo[3.2.0]hepta-1,5-dienes
Li, D., Rao, W., Tay, G. L., Ayers, B. J. & Chan, P. W. H., 2014, In : Journal of Organic Chemistry. 79, 23, p. 11301 - 11315 15 p.Research output: Contribution to journal › Article › Research › peer-review
Silica gel-mediated hydroamination/semipinacol rearrangement of 2-alkylaminophenylprop-1-yn-3-ols: synthesis of 2-oxindoles from alkynes and 1-(2-aminophenyl) ketones
Susanti, D., Ng, L. L. R. & Chan, P. W. H., 2014, In : Advanced Synthesis and Catalysis. 356, 2-3, p. 353 - 358 6 p.Research output: Contribution to journal › Article › Research › peer-review
Silver-catalyzed tandem hydroamination/hydroarylation of 1-(2-allylamino)phenyl-4-hydroxy-but-2-yn-1-ones to 1 '-allylspiro[indene-1,2 '-indolin]-3 '-ones
Mothe, S. R., Novianti, M. L., Ayers, B. J. & Chan, P. W. H., 2014, In : Organic Letters. 16, 16, p. 4110 - 4113 4 p.Research output: Contribution to journal › Article › Research › peer-review
Structure-based repurposing of FDA-approved drugs as inhibitors of NEDD8-activating enzyme
Zhong, H-J., Liu, L-J., Chan, D. S-H., Wang, H-M. D., Chan, P. W. H., Ma, D-L. E. & Leung, C-H. D., 2014, In : Biochimie. 102, 1, p. 211 - 215 5 p.Research output: Contribution to journal › Article › Research › peer-review
Synthesis of highly substituted indene derivatives by Bronsted acid catalyzed Friedel-Crafts reaction of homoallylic alcohols
Zhang, X., Teo, W. T., Rao, W., Ma, D-L. E., Leung, C-H. D. & Chan, P. W. H., 2014, In : Tetrahedron Letters. 55, 29, p. 3881 - 3884 4 p.Research output: Contribution to journal › Article › Research › peer-review
Ytterbium(III) triflate catalyzed annulation of propargylic 1,4-diols with aryl sulfonamides to give highly substituted pyrrole derivatives
Zhang, X., Teo, J. W., Ma, D-L. E., Leung, C-H. D. & Chan, P. W. H., 2014, In : Tetrahedron Letters. 55, 49, p. 6703 - 6707 5 p.Research output: Contribution to journal › Article › Research › peer-review
2013
1-(2′-Anilinyl)prop-2-yn-1-ol rearrangement for oxindole synthesis
Kothandaraman, P., Koh, B. Q., Limpanuparb, T., Hirao, H. & Chan, P. W. H., 4 Feb 2013, In : Chemistry - A European Journal. 19, 6, p. 1978-1985 8 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed cycloisomerization of 1,6-diyne carbonates and esters to 2,4a-dihydro-1H-fluorenes
Rao, W., Koh, M. J., Li, D., Hirao, H. & Chan, P. W. H., 2013, In : Journal of the American Chemical Society. 135, 21, p. 7926 - 7932 7 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed cycloisomerization of 1,7-enyne esters to structurally diverse cis-1,2,3,6-tetrahydropyridin-4-y1 ketones
Rao, W., Sally, U., Koh, M. J. & Chan, P. W. H., 2013, In : Journal of Organic Chemistry. 78, 7, p. 3183 - 3195 13 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed domino aminocyclization/1,3-sulfonyl migration of N-substituted N-sulfonyl-aminobut-3-yn-2-ols to 1-substituted 3-sulfonyl-1H-pyrroles
Teo, W. T., Rao, W., Koh, M. J. & Chan, P. W. H., 2013, In : Journal of Organic Chemistry. 78, 15, p. 7508 - 7517 10 p.Research output: Contribution to journal › Article › Research › peer-review
Metal-free synthesis of 1H-indole-2-carbaldehydes by N-iodosuccinimide-mediated cyclization of 1-(2 '-anilinyl)prop-2-yn-1-ols in water. A formal synthesis of (R)-calindol
Kothandaraman, P., Lauw, S. J. L. & Chan, P. W. H., 2013, In : Tetrahedron. 69, 35, p. 7471 - 7480 10 p.Research output: Contribution to journal › Article › Research › peer-review
Synthesis of (Z)-1,2-dihydro-1-tosylbenzo[b]azepin-3-ones by two-step, one-pot gold-catalyzed tandem heterocyclization/Petasis-Ferrier rearrangement of 2-(N-(prop-2-ynyl)-N-tosylamino)benzaldehydes
Sze, E. M. L., Koh, M. J., Tjia, Y. M., Rao, W. & Chan, P. W. H., 2013, In : Tetrahedron. 69, 26, p. 5558 - 5565 8 p.Research output: Contribution to journal › Article › Research › peer-review
2012
Bronsted acid-catalyzed cycloisomerization of but-2-yne-1,4-diols with or without 1,3-dicarbonyl compounds to tri- and tetrasubstituted furans
Mothe, S. R., Lauw, S. J. L., Kothandaraman, P. & Chan, P. W. H., 2012, In : Journal of Organic Chemistry. 77, 16, p. 6937 - 6947 11 p.Research output: Contribution to journal › Article › Research › peer-review
Copper(II) triflate catalyzed amination and aziridination of 2-alkyl substituted 1,3-dicarbonyl compounds
Ton, T. M. U., Tejo, C., Tiong, D. L. Y. & Chan, P. W. H., 2012, In : Journal of the American Chemical Society. 134, 17, p. 7344 - 7350 7 p.Research output: Contribution to journal › Article › Research › peer-review
Copper(II) triflate catalyzed amination of 1,3-dicarbonyl compounds
Ton, T. M. U., Himawan, F., Chang, J. W. W. & Chan, P. W. H., 17 Sep 2012, In : Chemistry - A European Journal. 18, 38, p. 12020-12027 8 p.Research output: Contribution to journal › Article › Research › peer-review
Gold-catalyzed cycloisomerization of 1,7-diyne benzoates to indeno[1,2-c]azepines and azabicyclo[4.2.0]octa-1(8),5-dines
Rao, W., Koh, M. J., Kothandaraman, P. & Chan, P. W. H., 2012, In : Journal of the American Chemical Society. 134, 26, p. 10811 - 10814 4 p.Research output: Contribution to journal › Article › Research › peer-review