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Research Output 2011 2019

2019

The TRPV4 Agonist GSK1016790A Regulates the Membrane Expression of TRPV4 Channels

Baratchi, S., Keov, P., Darby, W., Lai, A., Khoshmanesh, K., Thurgood, P., Vahidi, P., Ejendal, K. & McIntyre, P., 23 Jan 2019, In : Frontiers in Pharmacology. 10, 12 p., 6.

Research output: Contribution to journalArticleResearchpeer-review

Open Access
File
2018

Contractility measurements of human uterine smooth muscle to aid drug development

Arrowsmith, S., Keov, P., Muttenthaler, M. & Gruber, C. W., 26 Jan 2018, In : Journal of Visualized Experiments. 2018, 131, 12 p., e56639.

Research output: Contribution to journalArticleOtherpeer-review

Open Access
File

Discovery of peptide probes to modulate oxytocin-type receptors of insects

Keov, P., Liutkevičiute, Z., Hellinger, R., Clark, R. J. & Gruber, C. W., 1 Dec 2018, In : Scientific Reports. 8, 1, 7 p., 10020.

Research output: Contribution to journalArticleResearchpeer-review

Open Access
2017

Cyclotides isolated from an ipecac root extract antagonize the corticotropin releasing factor type 1 receptor

Fahradpour, M., Keov, P., Tognola, C., Perez-Santamarina, E., McCormick, P. J., Ghassempour, A. & Gruber, C. W., 25 Sep 2017, In : Frontiers in Pharmacology. 8, SEP, 14 p., 616.

Research output: Contribution to journalArticleResearchpeer-review

Open Access
File

Development of a human vasopressin V 1a -receptor antagonist from an evolutionary-related insect neuropeptide

Di Giglio, M. G., Muttenthaler, M., Harpsøe, K., Liutkeviciute, Z., Keov, P., Eder, T., Rattei, T., Arrowsmith, S., Wray, S., Marek, A., Elbert, T., Alewood, P. F., Gloriam, D. E. & Gruber, C. W., 1 Feb 2017, In : Scientific Reports. 7, 15 p., 41002.

Research output: Contribution to journalArticleResearchpeer-review

Open Access
File
2014

Molecular determinants of allosteric modulation at the M1 muscarinic acetylcholine receptor

Abdul Ridha, A., Lopez, L., Keov, P., Thal, D., Mistry, S. N., Sexton, P., Lane, J. R. D., Canals, M. & Christopoulos, A., 2014, In : Journal of Biological Chemistry. 289, 9, p. 6067 - 6079 13 p.

Research output: Contribution to journalArticleResearchpeer-review

Molecular mechanisms of bitopic ligand engagement with the M1 muscarinic acetylcholine receptor

Keov, P., Lopez, L., Devine, S., Valant, C., Lane, J. R. D., Scammells, P. J., Sexton, P. & Christopoulos, A., 2014, In : Journal of Biological Chemistry. 289, 34, p. 23817 - 23837 21 p.

Research output: Contribution to journalArticleResearchpeer-review

2011

Allosteric modulation of G protein-coupled receptors: A pharmacological perspective

Keov, P., Sexton, P. & Christopoulos, A., 2011, In : Neuropharmacology. 60, 1, p. 24 - 35 12 p.

Research output: Contribution to journalArticleResearchpeer-review