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Arthur Christopoulos

Professor

 https://orcid.org/0000-0003-4442-3294
1997 …2023
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Personal profile

Monash teaching commitment

  • Lectures to second year BPharm students in the Faculty of Pharmacy and Pharmaceutical Sciences
  • Lectures to third year BPharmSci students in the Faculty of Pharmacy and Pharmaceutical Sciences
  • Supervision of Honours students in Drug Discovery Biology
  • Supervision of PhD students in Drug Discovery Biology

Keywords

  • Analytical Pharmacology
  • Allosteric Modulation
  • Receptor Theory
  • Commentary: Drug Discovery
  • Pharmaceutical Research
  • Drug Side-Effects
  • Psychiatric Drugs
  • Supervision: Molecular Pharmacology
  • Drug Discovery
  • Receptors and Signal Transduction

Network Recent external collaboration on country level. Dive into details by clicking on the dots.

Projects 2004 2023

Adenosine A1 receptor modulation: Structure, dynamics & novel pharmacological interventions

Christopoulos, A., May, L. T., Imlach, W. L., Hill, S. & Scott, D.

1/01/18 → 31/12/22

Project: Research

NHMRC Equipment Grant - FLIPR Tetra high-throughput cellular screening system

Sexton, P., Christopoulos, A., Leach, K., Gregory, K. J., Veldhuis, N. A., Poole, D. P. & Langmead, C. J.

1/01/18 → 31/12/18

Project: Research

Collaborative Network to Define the Molecular Determinants of G Protein Coupled Receptor Clinical Efficacy

Christopoulos, A., Sexton, P. & Tobin, A.

1/11/16 → 31/10/21

Project: Research

Allosteric and Bitopic Ligands Acting at G Protein-Coupled Receptors

Scammells, P. J. & Christopoulos, A.

Australian Research Council (ARC), Monash University

1/01/16 → 31/12/18

Project: Research

The Janus face of G Protein-Coupled Receptors: Implications for Disease Mechanisms and Opportunities for Drug Discovery

Sexton, P., Bunnett, N., Christopoulos, A. & Summers, R. J.

National Health & Medical Research Council (NHMRC)

1/01/14 → 31/12/18

Project: Research

Research Output 1997 2018

Assessment of the molecular mechanisms of action of novel 4-phenylpyridine-2-one and 6-phenylpyrimidin-4-one allosteric modulators at the M1 muscarinic acetylcholine receptors

Van Der Westhuizen, E. T., Spathis, A., Khajehali, E., Jorg, M., Mistry, S. N., Capuano, B., Tobin, A. B., Sexton, P. M., Scammells, P. J., Valant, C. & Christopoulos, A. 24 Apr 2018 (Accepted/In press) In : Molecular Pharmacology. 50 p.

Research output: Contribution to journal › Article › Research › peer-review

Characterization of signalling and regulation of common calcitonin receptor splice variants and polymorphisms

Dal Maso, E., Just, R., Hick, C., Christopoulos, A., Sexton, P. M., Wootten, D. & Furness, S. G. B. 1 Feb 2018 In : Biochemical Pharmacology. 148, p. 111-129 19 p.

Research output: Contribution to journal › Article › Research › peer-review

Correspondence: Reply to 'Compound 17b and formyl peptide receptor biased agonism in relation to cardioprotective effects in ischaemia-reperfusion injury'

Qin, C. X., May, L. T., Sexton, P. M., DeBono, A. J., Baell, J. B., Christopoulos, A. & Ritchie, R. H. 1 Dec 2018 In : Nature Communications. 9, 1, 4 p., 530

Research output: Contribution to journal › Letter › Other › peer-review

Open Access
File

Differential engagement of polar networks in the glucagon-like peptide 1 receptor by endogenous variants of the glucagon-like peptide 1

Furness, S. G. B., Christopoulos, A., Sexton, P. M. & Wootten, D. 1 Oct 2018 In : Biochemical Pharmacology. 156, p. 223-240 18 p.

Research output: Contribution to journal › Article › Research › peer-review

Dominant Negative G Proteins Enhance Formation and Purification of Agonist-GPCR-G Protein Complexes for Structure Determination

Liang, Y-L., Zhao, P., Draper-Joyce, C. J., Baltos, J-A., Glukhova, A., Truong, T. T., May, L. T., Christopoulos, A., Wootten, D., Sexton, P. & Furness, S. 26 Jul 2018 (Accepted/In press) In : ACS Pharmacology and Translational Sciences. 9 p.

Research output: Contribution to journal › Article › Research › peer-review

Open Access

Activities 2011 2011

  • 1 Submissions to industry or govt committees, commissions and inquiries

Theme Leader

Christopoulos, A. (Member)
10 Nov 2011

Activity: Submissions to industry or govt committees, commissions and inquiries