Research Output 1977 2019

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2009
76 Citations (Scopus)

Kinetic studies of AKR1B10, human aldose reductase-like protein: Endogenous substrates and inhibition by steroids

Endo, S., Matsunaga, T., Mamiya, H., Ohta, C., Soda, M., Kitade, Y., Tajima, K., Zhao, H-T., El-Kabbani, O. & Hara, A., 2009, In : Archives of Biochemistry and Biophysics. 487, 1, p. 1 - 9 9 p.

Research output: Contribution to journalArticleResearchpeer-review

10 Citations (Scopus)

Linear and convergent approaches to 2-substituted adenosine-5 '-N-alkylcarboxamides

Foitzik, R., Devine, S., Hausler, N. E. & Scammells, P. J., 2009, In : Tetrahedron. 65, 43, p. 8851 - 8857 7 p.

Research output: Contribution to journalArticleResearchpeer-review

12 Citations (Scopus)

Molecular determinants for the stereospecific reduction of 3-ketosteroids and reactivity towards all-trans-retinal of a short-chain dehydrogenase/reductase (DHRS4)

Endo, S., Maeda, S., Matsunaga, T., Dhagat, U., El-Kabbani, O., Tanaka, N., Nakamura, K. T., Tajima, K. & Hara, A., 2009, In : Archives of Biochemistry and Biophysics. 481, 2, p. 183 - 190 8 p.

Research output: Contribution to journalArticleResearchpeer-review

54 Citations (Scopus)

Molecular docking of carbohydrate ligands to antibodies: Structural validation against crystal structures

Agostino, M. J., Jene, C., Boyle, T. P., Ramsland, P. A. & Yuriev, E., 2009, In : Journal of Chemical Information and Modeling. 49, 12, p. 2749 - 2760 12 p.

Research output: Contribution to journalArticleResearchpeer-review

25 Citations (Scopus)

Molecular Dynamics of Poly(L-lysine) Dendrimers with Naphthalene Disulfonate Caps

Roberts, B. P., Scanlon, M., Krippner, G. Y. & Chalmers, D. K., 2009, In : Macromolecules. 42, 7, p. 2775 - 2783 9 p.

Research output: Contribution to journalArticleResearchpeer-review

18 Citations (Scopus)

Molecular dynamics of variegated polyamide dendrimers

Roberts, B. P., Krippner, G. Y., Scanlon, M. & Chalmers, D. K., 2009, In : Macromolecules. 42, 7, p. 2784 - 2794 11 p.

Research output: Contribution to journalArticleResearchpeer-review

24 Citations (Scopus)

New macrocyclic terbium(III) complex for use in RNA footprinting experiments

Belousoff, M. J., Ung, P., Forsyth, C. M., Tor, Y., Spiccia, L. & Graham, B., 2009, In : Journal of the American Chemical Society. 131, p. 1106 - 1114 9 p.

Research output: Contribution to journalArticleResearchpeer-review

2 Citations (Scopus)

NMR assignment of prespore specific antigen-a cell surface adhesion glycoprotein from Dictyostelium discoideum

Swarbrick, J. D., Cubeddu, L., Ball, G. E., Curmi, P. MG., Gooley, A. A., Williams, K. L. & Mabbutt, B., 2009, In : Biomolecular NMR Assignments. 3, 1, p. 1 - 3 3 p.

Research output: Contribution to journalArticleResearchpeer-review

Novel thrombopoietin mimics for haemopoietic stem cell expansion

Haylock, DN., Andrade, J., White, J., Nilsson, SK., Meagher, L., Cableswki, T., Schwab, K., Tarasova, A., Condie, G., Riches, A. & Winkler, D. A., 2009, In : Experimental Hematology. 37, 9 Suppl 1

Research output: Contribution to journalArticleResearchpeer-review

83 Citations (Scopus)

Phosphonium ionic liquids: design, synthesis and evaluation of biodegradability

Atefi, F., Garcia, M. T., Singer, R. D. & Scammells, P. J., 2009, In : Green Chemistry. 11, 10, p. 1595 - 1604 10 p.

Research output: Contribution to journalArticleResearchpeer-review

48 Citations (Scopus)

Potent and selective inhibition of the tumor marker AKR1B10 by bisdemethoxycurcumin: Probing the active site of the enzyme with molecular modeling and site-directed mutagenesis

Matsunaga, T., Endo, S., Soda, M., Zhao, H-T., El-Kabbani, O., Tajima, K. & Hara, A., 2009, In : Biochemical and Biophysical Research Communications. 389, 1, p. 128 - 132 5 p.

Research output: Contribution to journalArticleResearchpeer-review

5 Citations (Scopus)

Predictive mesoscale network model of cell fate decisions during C. elegans embryogenesis

Winkler, D. A., Burden, F. R. & Halley, J. D., 2009, In : Artificial Life. 15, 4, p. 411-421 11 p.

Research output: Contribution to journalArticleResearchpeer-review

15 Citations (Scopus)

Probing the fibrate binding specificity of rat liver fatty acid binding protein

Chuang, S., Velkov, T., Horne, H. J., Wielens, J., Chalmers, D. K., Porter, C. J. & Scanlon, M., 2009, In : Journal of Medicinal Chemistry. 52, 17, p. 5344 - 5355 12 p.

Research output: Contribution to journalArticleResearchpeer-review

25 Citations (Scopus)

RAFT-mediated polymerization of styrene in readily biodegradable ionic liquids

Johnston-Hall, G., Harjani, J. R., Scammells, P. J. & Monteiro, M. J., 2009, In : Macromolecules. 42, 5, p. 1604 - 1609 5 p.

Research output: Contribution to journalArticleResearchpeer-review

7 Citations (Scopus)

Reaction pathways to 2-aminothiophenes and thiophene-3-carbonitriles

Aurelio, L., Flynn, B. L. & Scammells, P. J., 2009, In : Australian Journal of Chemistry. 62, 5, p. 402 - 406 5 p.

Research output: Contribution to journalArticleResearchpeer-review

18 Citations (Scopus)

Structural biology of carbohydrate xenoantigens

Yuriev, E., Agostino, M. J., Farrugia, W., Christiansen, D., Sandrin, M. S. & Ramsland, P. A., 2009, In : Expert Opinion on Biological Therapy. 9, 8, p. 1017 - 1029 13 p.

Research output: Contribution to journalArticleResearchpeer-review

4 Citations (Scopus)

Structure/function analysis of a critical disulfide bond in the active site of l-xylulose reductase

Zhao, H-T., Endo, S., Ishikura, S., Chung, R. P-T., Hogg, P. J., Hara, A. & El-Kabbani, O., 2009, In : Cellular and Molecular Life Sciences. 66, 9, p. 1570 - 1579 10 p.

Research output: Contribution to journalArticleResearchpeer-review

18 Citations (Scopus)

Structure and dynamics of glyceride lipid formulations, with propylene glycol and water

Warren, D., Chalmers, D. K. & Pouton, C. W., 2009, In : Molecular Pharmaceutics. 6, 2, p. 604 - 614 11 p.

Research output: Contribution to journalArticleResearchpeer-review

25 Citations (Scopus)

Structure and function of the oxidoreductase DsbA1 from Neisseria meningitidis

Vivian, J., Scoullar, J., Rimmer, K., Bushell, S. R., Beddoe, T. C., Wilce, M. C. J., Byres, E., Boyle, T. P., Doak, B. C., Simpson, J. S., Graham, B., Heras, B., Kahler, C. M., Rossjohn, J. & Scanlon, M., 2009, In : Journal of Molecular Biology. 394, 5, p. 931 - 943 13 p.

Research output: Contribution to journalArticleResearchpeer-review

22 Citations (Scopus)

Structure-guided design, synthesis, and evaluation of salicylic acid-based inhibitors targeting a selectivity pocket in the active site of human 20alpha-hydroxysteroid dehydrogenase (AKR1C1)

El-Kabbani, O., Scammells, P. J., Gosling, J. I., Dhagat, U., Endo, S., Matsunaga, T., Soda, M. & Hara, A., 2009, In : Journal of Medicinal Chemistry. 52, 10, p. 3259 - 3264 6 p.

Research output: Contribution to journalArticleResearchpeer-review

25 Citations (Scopus)

Structure of granzyme C reveals an unusual mechanism of protease autoinhibition

Kaiserman, D., Buckle, A. M., Van Damme, P., Irving, J. A., Law, R. H. P., Matthews, A. Y., Bashtannyk-Puhalovich, T. A., Langendorf, C., Thompson, P., Vandekerckhove, J., Gevaert, K., Whisstock, J. C. & Bird, P. I., 2009, In : Proceedings of the National Academy of Sciences. 106, 14, p. 5587 - 5592 6 p.

Research output: Contribution to journalArticleResearchpeer-review

2 Citations (Scopus)

Structure of the G225P/G226P mutant of mouse 3(17)alpha-hydroxysteroid dehydrogenase (AKR1C21) ternary complex: Implications for the binding of inhibitor and substrate

Dhagat, U., Endo, S., Mamiya, H., Hara, A. & El-Kabbani, O., 2009, In : Acta Crystallographica Section D: Biological Crystallography. 65, 3, p. 257 - 265 9 p.

Research output: Contribution to journalArticleResearchpeer-review

8 Citations (Scopus)

Synthesis and evaluation of dithiolethiones as novel cyclooxygenase inhibitors

Zanatta, S. D., Manallack, D. T., Jarrott, B. & Williams, S. J., 2009, In : Bioorganic and Medicinal Chemistry Letters. 19, 2, p. 459 - 461 3 p.

Research output: Contribution to journalArticleResearchpeer-review

8 Citations (Scopus)

Synthesis and preliminary screening of novel indole-3-methanamines as 5-HT4 receptor ligands

Hanna-Elias, A., Manallack, D. T., Berque-Bestel, I., Irving, H. R., Coupar, I. M. & Iskander, M. N., 2009, In : European Journal of Medicinal Chemistry. 44, 7, p. 2952 - 2959 8 p.

Research output: Contribution to journalArticleResearchpeer-review

6 Citations (Scopus)

Synthesis of quinoline derivatives as 5-HT4 receptor ligands

Hanna-Elias, A., Manallack, D. T., Berque-Bestel, I., Irving, H. R., Coupar, I. M. & Iskander, M. N., 2009, In : Australian Journal of Chemistry. 62, 2, p. 150 - 156 7 p.

Research output: Contribution to journalArticleResearchpeer-review

40 Citations (Scopus)

The acid-base profile of a contemporary set of drugs: implications for drug discovery

Manallack, D. T., 2009, In : SAR and QSAR in Environmental Research. 20, 7-8, p. 611 - 655 45 p.

Research output: Contribution to journalArticleResearchpeer-review

14 Citations (Scopus)

The effects of exosite occupancy on the substrate specificity of thrombin

Ng, N. M-Y., Quinsey, N. S., Matthews, A. Y., Kaiserman, D., Wijeyewickrema, L. C., Bird, P. I., Thompson, P. E. & Pike, R. N., 2009, In : Archives of Biochemistry and Biophysics. 489, 1-2, p. 48 - 54 7 p.

Research output: Contribution to journalArticleResearchpeer-review

10 Citations (Scopus)

The identification and optimisation of novel and selective diamide neuropeptide Y Y2 receptor antagonists

Lunniss, G. E., Barnes, A. A., Barton, N., Biagetti, M., Bianchi, F., Blowers, S. M., Caberlotto, L., Emmons, A., Holmes, I. P., Montanari, D., Norris, R., Walters, D. J. & Watson, S. P., 2009, In : Bioorganic and Medicinal Chemistry Letters. 19, 15, p. 4022 - 4025 4 p.

Research output: Contribution to journalArticleResearchpeer-review

12 Citations (Scopus)

The identification of beta-hydroxy carboxylic acids as selective MMP-12 inhibitors.

Holmes, I. P., Gaines, S., Watson, S. P., Lorthioir, O., Walker, A., Baddeley, S. J., Herbert, S., Egan, D., Convery, M. A., Singh, O. M. P., Gross, J. W., Strelow, J. M., Smith, R. H., Amour, A. J., Brown, D. & Stephen, M. L., 2009, In : Bioorganic and Medicinal Chemistry Letters. 19, 19, p. 5760 - 5763 4 p.

Research output: Contribution to journalArticleResearchpeer-review

12 Citations (Scopus)

Thermodynamics of lipophilic drug binding to intestinal fatty acid binding protein and permeation across membranes

Velkov, T., 6 Apr 2009, In : Molecular Pharmaceutics. 6, 2, p. 557-570 14 p.

Research output: Contribution to journalArticleResearchpeer-review

41 Citations (Scopus)

The Structure of the Bacterial Oxidoreductase Enzyme DsbA in Complex with a Peptide Reveals a Basis for Substrate Specificity in the Catalytic Cycle of DsbA Enzymes

Paxman, J. J., Borg, N., Horne, H. J., Thompson, P., Chin, K. Y., Sharma, P., Simpson, J. S., Wielens, J., Piek, S., Kahler, C. M., Sakellaris, H., Pearce, M. C., Bottomley, S. P., Rossjohn, J. & Scanlon, M., 2009, In : Journal of Biological Chemistry. 284, 26, p. 17835 - 17845 11 p.

Research output: Contribution to journalArticleResearchpeer-review

1 Citation (Scopus)

The Use of Tripeptides for Lead Discovery of 5-HT4 Receptor Ligands

Hanna-Elias, A., Thompson, P., Manallack, D. T., Irving, H. R., Coupar, I. M., Berque-Bestel, I. & Iskander, M. N., 2009, In : Protein and Peptide Letters. 16, 7, p. 805 - 809 5 p.

Research output: Contribution to journalArticleResearchpeer-review

60 Citations (Scopus)

Total Synthesis of the Potent Anticancer Aglaia Metabolites (-)-Silvestrol and (-)-Episilvestrol and the Active Analogue (-)-4-Desmethoxyepisilvestrol

Adams, T. E., El Sous, M., Hawkins, B. C., Hirner, S., Holloway, G. A., Khoo, M. L., Owen, D. J., Savage, G. P., Scammells, P. J. & Rizzacasa, M. A., 2009, In : Journal of the American Chemical Society. 131, 4, p. 1607 - 1616 10 p.

Research output: Contribution to journalArticleResearchpeer-review

2010
466 Citations (Scopus)

10-year stroke prevention after successful carotid endarterectomy for asymptomatic stenosis (ACST-1): A multicentre randomised trial

Halliday, A., Harrison, M., Hayter, E., Kong, X., Mansfield, A., Marro, J., Pan, H., Peto, R., Potter, J., Rahimi, K., Rau, A., Robertson, S., Streifler, J., Thomas, D., Cooper, M. E., MacKay, M., Wood, J., Christopoulos, G., Pereira, M. C., Blomstrand, C. & 205 others, Forssell, C., Potemkowski, A., Skiöldebrand, C., Stoor, P., Blomqvist, M., Calander, M., Forssell, C., Lundgren, F., Almqvist, H., Norgren, L., Norrving, B., Ribbe, E., Thörne, J., Gottsäter, A., Mätzsch, T., Nilsson, M. E., Forssell, C., Lonsson, M., Lundgren, F., Stahre, B., Norgren, L., Stenberg, B., Konrad, P., Jarl, L., Lundqvist, L., Olofsson, P., Rosfors, S., Skiöldebrand, C., Swedenborg, J., Takolander, R., Bergqvist, D., Ljungman, C., Pärsson, H., Kniemeyer, H. W., Widmer, M. K., Kuster, R., Kaiser, R., Nagel, W., Sege, D., Weder, B., Nie, J., Doelman, J., Yilmaz, N. K., Buth, J., Stultiens, G., Boiten, J., Boon, R. A., van der Linden, F., Busman, D. C., Sinnige, H. A. W., Yo, T. I., de Borst, G. J., Eikelboom, B. C., Kappelle, L. J., Tovar-Moll, F., van Reedt Dortland, R. W. H., Westra, T. E., Jaber, H., Manaa, J., Meftah, R. B., Nabil, B. R., Sraieb, T., Bateman, E. D., Budd, J., Horrocks, M., Kivela, M., Shaw, L., Walker, R., D'Sa, A. A. B. B., Simms, M. S., Baird, R., Campbell, M., Cole, S., Ferguson, I. T., Lamont, P. J., Mitchell, D., Sassano, A., Smith, F. C. T., Blake, K. L., Kirkpatrick, P. J., Martin, P., Turner, P. C., Clegg, J. F., Crosley, M., Hall, J., de Cossart, L., Edwards, P., Fletcher, D., Stigger-Rosser, E., McCollum, P. T., Davidson, D., Levison, R., Bradbury, A. W., Chalmers, R. T. A., Dennis, M., Murie, J. A., Ruckley, C. V., Sandercock, P., Campbell, W. B., Frankel, T., Gardner-Thorpe, C., Gutowski, N., Hardie, R. E., Honan, W., Niblett, P., Peters, A., Ridler, B., Thompson, J. F., Bone, I., Welch, G. C., Grocott, E. C., Overstall, P., Aldoori, M. I., Dafalla, B. E. A., Bryce, J., Clarke, C., McCollum, P. T., Ming, A-X., Wilkinson, A. R., Bamford, J., Berridge, D., Scott, J., Abbott, R. J., Naylor, R., Harris, P., Humphrey, Q. P. C., Adiseshiah, M., Aukett, M., Baker, D., Bishop, C. C. R., Boutin, A., Brown, M., Burke, P., Burnand, K. G., Colchester, A., Coward, L., Davies, A. H., Espasandin, M., Giddings, A. E. B., Hamilton, G., Judge, C., Kakkos, S. K., McGuiness, C., Morris-Vincent, P., Nicolaides, A. N., Padayachee, T. S., Riordan, H., Sullivan, E., Taylor, P., Thompson, M., Wolfe, J. H. N., McCollum, C. N., O'Neill, P. A., Welsh, S., Barnes, J., Cleland, P., Davis, M., Gholkar, A., Jones, R., Jaykishnam, V., Mendelow, A. D., O'Connell, J. E., Siddique, M. S. S., Stansby, G., Vivar, R., Ashley, S., Cosgrove, C., Gibson, J., Wilkins, D. C., Chant, A. D. B., Frankel, J., Shearman, C. P., Williams, J., Hall, G., Holdsworth, R., Davies, J. N., McLean, B., Woodburn, K. R., Brown, G., Curley, P., Loizou, L., Chaturvedi, S., Diaz, R. F., Radak, D., Todorovic, P. R., Kamugasha, D., Baxter, A., Berry, C., Burrett, J., Collins, R., Crowther, M. J., Davies, C., Farrell, B., Godwin, J., Gray, R., Harwood, C., Hirt, L., Hope, C., Knight, S., Lay, M., Munday, A., Murawska, A., Peto, C. G., Radley, A. & Richards, S., 25 Sep 2010, In : The Lancet. 376, 9746, p. 1074-1084 11 p.

Research output: Contribution to journalArticleResearchpeer-review

24 Citations (Scopus)

An efficient synthesis of (+-)-frondosin B using a Stille-Heck reaction sequence

Masters, K-S. & Flynn, B. L., 2010, In : Organic and Biomolecular Chemistry. 8, 6, p. 1290 - 1292 3 p.

Research output: Contribution to journalArticleResearchpeer-review

22 Citations (Scopus)

Antiviral agents 2. Synthesis of trimeric naphthoquinone analogues of conocurvone and their antiviral evaluation against HIV

Crosby, I., Bourke, D., Jones, E., De Bruyn, P., Rhodes, D., Vandergraaff, N., Cox, S., Coates, J. & Robertson, A., 2010, In : Bioorganic & Medicinal Chemistry. 18, 17, p. 6442 - 6450 9 p.

Research output: Contribution to journalArticleResearchpeer-review

35 Citations (Scopus)

A reductive-coupling plus Nazarov cyclization sequence in the asymmetric synthesis of five-membered carbocycles

Kerr, D., White, J. & Flynn, B., 2010, In : Journal of Organic Chemistry. 75, 21, p. 7073 - 7084 12 p.

Research output: Contribution to journalArticleResearchpeer-review

2 Citations (Scopus)

Backbone and side chain 1H, 15N and 13C assignments for the oxidised and reduced forms of the oxidoreductase protein DsbA from Staphylococcus aureus

Williams, M. L., Chalmers, D. K., Martin, J. L. & Scanlon, M., Apr 2010, In : Biomolecular NMR Assignments. 4, 1, p. 25 - 28 4 p.

Research output: Contribution to journalArticleResearchpeer-review

3 Citations (Scopus)

Binding mode prediction of PDE4 inhibitors: a comparison of modelling methods

Neale, D., Thompson, P., White, P., Chalmers, D., Yuriev, E. & Manallack, D., 2010, In : Australian Journal of Chemistry. 63, 3, p. 396 - 404 9 p.

Research output: Contribution to journalArticleResearchpeer-review

61 Citations (Scopus)

BNC105: A novel tubulin polymerization inhibitor that selectively disrupts tumor vasculature and displays single-agent antitumor efficacy

Kremmidiotis, G., Leske, A., Lavranos, T., Beaumont, D., Gasic, J., Hall, A., O'Callaghan, M., Matthews, C. & Flynn, B., 2010, In : Molecular Cancer Therapeutics. 9, 6, p. 1562 - 1573 12 p.

Research output: Contribution to journalArticleResearchpeer-review

21 Citations (Scopus)

Characterization of the DsbA oxidative folding catalyst from Pseudomonas aeruginosa reveals a highly oxidizing protein that binds small molecules

Shouldice, S., Heras, B., Jarrott, R., Sharma, P., Scanlon, M. & Martin, J., 2010, In : Antioxidants and Redox Signaling. 12, 8, p. 921 - 931 11 p.

Research output: Contribution to journalArticleResearchpeer-review

58 Citations (Scopus)

Chromene-3-carboxamide derivatives discovered from virtual screening as potent inhibitors of the tumour maker, AKR1B10

Endo, S., Matsunaga, T., Kuwata, K., Zhao, H-T., El-Kabbani, O., Kitade, Y. & Hara, A., 2010, In : Bioorganic & Medicinal Chemistry. 18, 7, p. 2485 - 2490 6 p.

Research output: Contribution to journalArticleResearchpeer-review

16 Citations (Scopus)

Comparison of NMR and crystal structures highlights conformational isomerism in protein active sites

Serrano, P., Serrano, P., Pedrini, B., Pedrini, B., Geralt, M., Jaudzems, K., Jaudzems, K., Mohanty, B., Mohanty, B., Horst, R., Horst, R., Herrmann, T., Elsliger, M. A., Elsliger, M. A., Wilson, I. A., Wilson, I. A., Wilson, I. A., Wüthrich, K., Wüthrich, K., Wüthrich, K. & 1 others, Wüthrich, K., 1 Oct 2010, In : Acta Crystallographica. Section F: Structural Biology Communications. 66, 10, p. 1393-1405 13 p.

Research output: Contribution to journalArticleResearchpeer-review

6 Citations (Scopus)

Crystallization and preliminary X-ray analysis of 6 - Hydroxymethyl-7,8- dihydropterin pyrophosphokinase from Staphylococcus aureus

Chhabra, S., Newman, J., Peat, T. S., Fernley, R. T., Caine, J., Simpson, J. S. & Swarbrick, J. D., 2010, In : Acta Crystallographica. Section F: Structural Biology Communications. 66, 5, p. 575 - 578 4 p.

Research output: Contribution to journalArticleResearchpeer-review

38 Citations (Scopus)

Crystal structure of the HIV-1 integrase core domain in complex with sucrose reveals details of an allosteric inhibitory binding site

Wielens, J., Headey, S., Jeevarajah, D., Rhodes, D., Deadman, J., Chalmers, D., Scanlon, M. & Parker, M., 2010, In : FEBS Letters. 584, 8, p. 1455 - 1462 8 p.

Research output: Contribution to journalArticleResearchpeer-review

33 Citations (Scopus)

Delineating the mode of action of adenosine A1 receptor allosteric modulators

Valant, C., Aurelio, L., Urmaliya, V., White, P., Scammells, P., Sexton, P. & Christopoulos, A., 2010, In : Molecular Pharmacology. 78, 3, p. 444 - 455 12 p.

Research output: Contribution to journalArticleResearchpeer-review

32 Citations (Scopus)

Developing an anion host for lipid A binding and antibacterial activity

Henderson, L. C., Li, J., Nation, R. L., Velkov, T. & Pfeffer, F. M., 2010, In : Chemical Communications. 46, p. 3197 - 3199 3 p.

Research output: Contribution to journalArticleResearchpeer-review

23 Citations (Scopus)

Effects of conformational restriction of 2-amino-3-benzoylthiophenes on A1 adenosine receptor modulation

Aurelio, L., Valant, C., Flynn, B., Sexton, P., White, J., Christopoulos, A. & Scammells, P., 2010, In : Journal of Medicinal Chemistry. 53, p. 6550 - 6559 10 p.

Research output: Contribution to journalArticleResearchpeer-review

1 Citation (Scopus)

Factorizing the role of a critical leucine residue in the binding of substrate to human 20alpha-hydroxysteroid dehydrogenase (AKR1C1): Molecular modeling and kinetic studies of the Leu308Val mutant enzyme

Dhagat, U., Endo, S., Soda, M., Hara, A. & El-Kabbani, O., 2010, In : Bioorganic and Medicinal Chemistry Letters. 20, 17, p. 5274 - 5276 3 p.

Research output: Contribution to journalArticleResearchpeer-review